Research Article
Open Access
Discovery of a cofactor-independent inhibitor of Mycobacterium tuberculosis InhA
Yi Xia, Yasheen Zhou, David S Carter, Matthew B McNeil, Wai Choi, Jason Halladay, Pamela W Berry, Weimin Mao, Vincent Hernandez, Theresa O'Malley, Aaron Korkegian, Bjorn Sunde, Lindsay Flint, Lisa K Woolhiser, Michael S Scherman, Veronica Gruppo, Courtney Hastings, Gregory T Robertson, Thomas R Ioerger, Jim Sacchettini, Peter J Tonge, Anne J Lenaerts, View ORCID ProfileTanya Parish Correspondence email, MRK Alley
Yi Xia
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Yasheen Zhou
1Anacor Pharmaceuticals, Palo Alto, CA, USA
David S Carter
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Matthew B McNeil
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
Wai Choi
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Jason Halladay
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Pamela W Berry
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Weimin Mao
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Vincent Hernandez
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Theresa O'Malley
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
Aaron Korkegian
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
Bjorn Sunde
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
Lindsay Flint
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
Lisa K Woolhiser
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Michael S Scherman
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Veronica Gruppo
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Courtney Hastings
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Gregory T Robertson
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Thomas R Ioerger
4Texas A&M University, College Station, TX, USA
Jim Sacchettini
4Texas A&M University, College Station, TX, USA
Peter J Tonge
5Institute of Chemical Biology and Drug Discovery, Departments of Chemistry and Radiology, Stony Brook University, Stony Brook, NY, USA
Anne J Lenaerts
3Mycobacteria Research Laboratories, Department of Microbiology, Immunology, and Pathology, Colorado State University, Fort Collins, CO, USA
Tanya Parish
2TB Discovery Research, Infectious Disease Research Institute, Seattle, WA, USA
MRK Alley
1Anacor Pharmaceuticals, Palo Alto, CA, USA
Published 1 June 2018. DOI: 10.26508/lsa.201800025
Direct inhibition of Mycobacterium tuberculosis InhA
Yi Xia, Yasheen Zhou, David S Carter, Matthew B McNeil, Wai Choi, Jason Halladay, Pamela W Berry, Weimin Mao, Vincent Hernandez, Theresa O'Malley, Aaron Korkegian, Bjorn Sunde, Lindsay Flint, Lisa K Woolhiser, Michael S Scherman, Veronica Gruppo, Courtney Hastings, Gregory T Robertson, Thomas R Ioerger, Jim Sacchettini, Peter J Tonge, Anne J Lenaerts, Tanya Parish, MRK Alley
Life Science Alliance Jun 2018, 1 (3) e201800025; DOI: 10.26508/lsa.201800025
Direct inhibition of Mycobacterium tuberculosis InhA
Yi Xia, Yasheen Zhou, David S Carter, Matthew B McNeil, Wai Choi, Jason Halladay, Pamela W Berry, Weimin Mao, Vincent Hernandez, Theresa O'Malley, Aaron Korkegian, Bjorn Sunde, Lindsay Flint, Lisa K Woolhiser, Michael S Scherman, Veronica Gruppo, Courtney Hastings, Gregory T Robertson, Thomas R Ioerger, Jim Sacchettini, Peter J Tonge, Anne J Lenaerts, Tanya Parish, MRK Alley
Life Science Alliance Jun 2018, 1 (3) e201800025; DOI: 10.26508/lsa.201800025
In this Issue
Volume 1, No. 3
June 2018
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